SCHEMBL6601667

SCHEMBL6601667

CS(=O)(=O)c1cccc(-c2cnn(Cc3ccccc3)c(=O)c2Br)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.61
PTGS1 P23219 6/20 0.61
MET P08581 2/20 0.43
NTRK1 P04629 1/20 0.43
PIM1 P11309 1/20 0.43
FGFR1 P11362 1/20 0.43
MAP2K2 P36507 1/20 0.43
FLT3 P36888 1/20 0.43
MAPK8 P45983 1/20 0.43
GSK3B P49841 1/20 0.43
NTRK3 Q16288 1/20 0.43
ALK Q9UM73 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
KCNH2 Q12809 1/20 0.43
PFKFB3 Q16875 1/20 0.41
DRD2 P14416 1/20 0.41
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601380 0.88 PTGS2 (0.79) PTGS2PTGS1
SCHEMBL6601664 0.87 PTGS2 (0.75) PTGS2PTGS1PFKFB3
SCHEMBL6600842 0.83 PTGS2 (0.81) PTGS2PTGS1
SCHEMBL6606371 0.82 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL6601421 0.82 PTGS2 (0.59) PTGS2PTGS1METNTRK1PIM1
SCHEMBL6602267 0.82 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL6602110 0.82 PTGS2 (0.66) PTGS2PTGS1METNTRK1PIM1
SCHEMBL6600014 0.81 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL6605804 0.81 PTGS2 (0.47) PTGS2PTGS1PFKFB3
SCHEMBL6605506 0.81 PTGS2 (0.82) PTGS2PTGS1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975604-B1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 2004-07-21 EP disclosed
EP-0975604-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 Merck Frosst Canada & Co. (CA) 2000-02-02 EP disclosed
US-6004960-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION MERCK FROSST CANADA, INC. (CA) 1999-12-21 US disclosed
WO-1998041511-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 1998-09-24 WO disclosed