SCHEMBL6601801

SCHEMBL6601801

O=C(NS(=O)(=O)c1ccc(-c2ccc3c(c2)CCC(CNC[C@@H](O)c2cccnc2)O3)cc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 16/20 0.47
PTGS2 P35354 4/20 0.43
ADRB1 P08588 10/20 0.42
ADRB2 P07550 6/20 0.42
PTGS1 P23219 2/20 0.41
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6284152 1.00 ADRB3 (0.47) ADRB3PTGS2ADRB1ADRB2PTGS1
SCHEMBL6284156 1.00 ADRB3 (0.47) ADRB3PTGS2ADRB1ADRB2PTGS1
SCHEMBL6279899 0.94 ADRB3 (0.45) ADRB3PTGS2ADRB1ADRB2
SCHEMBL6279905 0.94 ADRB3 (0.45) ADRB3PTGS2ADRB1ADRB2
SCHEMBL6284449 0.92 ADRB3 (0.44) ADRB3ADRB1ADRB2
SCHEMBL6284439 0.92 ADRB3 (0.44) ADRB3ADRB1ADRB2
SCHEMBL6283986 0.91 PTGS2 (0.46) ADRB3PTGS2ADRB1ADRB2
SCHEMBL6283980 0.91 PTGS2 (0.46) ADRB3PTGS2ADRB1ADRB2
SCHEMBL6277922 0.90 ADRB3 (0.42) ADRB3PTGS2ADRB1ADRB2PTGS1
SCHEMBL6277919 0.90 ADRB3 (0.42) ADRB3PTGS2ADRB1ADRB2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389202-B1 2,6-SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER PHARMACEUTICALS CORP (US) 2004-09-29 EP claimed