SCHEMBL6601976

SCHEMBL6601976

Cn1ncc(-c2ccc(S(C)(=O)=O)cc2)c(-c2ccccc2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 1.00
PTGS1 P23219 8/20 0.68
ITGB1 P05556 1/20 0.58
ITGA4 P13612 1/20 0.58
ITGB7 P26010 1/20 0.58
ALOX5 P09917 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8381355 0.87 PTGS2 (0.76) PTGS2PTGS1ITGB1ITGA4ITGB7
SCHEMBL6601979 0.87 PTGS2 (0.77) PTGS2PTGS1ITGB1ITGA4ITGB7
SCHEMBL6603152 0.84 PTGS2 (1.00) PTGS2PTGS1ALOX5
SCHEMBL6601509 0.83 PTGS2 (0.71) PTGS2PTGS1ITGB1ITGA4ITGB7
SCHEMBL6601374 0.81 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6601032 0.79 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6599964 0.78 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL4186362 0.78 PTGS2 (0.83) PTGS2PTGS1
SCHEMBL4191548 0.78 PTGS2 (0.86) PTGS2PTGS1
SCHEMBL6601027 0.77 PTGS2 (0.79) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004960-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION MERCK FROSST CANADA, INC. (CA) 1999-12-21 US claimed
EP-0975604-B1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 2004-07-21 EP disclosed
EP-0975604-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 Merck Frosst Canada & Co. (CA) 2000-02-02 EP disclosed
US-6004960-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION MERCK FROSST CANADA, INC. (CA) 1999-12-21 US disclosed
WO-1998041511-A1 PYRIDAZINONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 1998-09-24 WO disclosed