SCHEMBL6602371

SCHEMBL6602371

CNC(=O)c1noc(C(Cc2ccc3ccccc3c2)N(C)C(=O)C(N)Cc2ccc3ccccc3c2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 3/20 0.40
MC3R P41968 3/20 0.40
MC5R P33032 2/20 0.40
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
SLC7A11 Q9UPY5 1/20 0.38
ZAP70 P43403 3/20 0.37
SRC P12931 2/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
GHSR Q92847 1/20 0.37
DPP4 P27487 1/20 0.36
MME P08473 2/20 0.36
TPH1 P17752 2/20 0.36
SLC7A5 Q01650 1/20 0.36
TACR1 P25103 1/20 0.36
ACE P12821 1/20 0.35
MC1R Q01726 1/20 0.35
F2 P00734 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602122 0.97 MC4R (0.42) MC4RMC3RMC5RMMP9MMP8
SCHEMBL27477310 0.89 MC4R (0.44) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6601903 0.89 MC4R (0.44) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6600540 0.89 MC4R (0.42) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6601083 0.88 MC4R (0.41) MC4RMC3RMC5RSLC7A11GHSR
SCHEMBL3728182 0.86 MC4R (0.43) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6317958 0.85 MC4R (0.43) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6613846 0.85 MC4R (0.43) MC4RMC3RMC5RMMP9MMP8
SCHEMBL6600886 0.85 MMP2 (0.42) MC4RMC3RMC5RMMP9MMP8
SCHEMBL4282449 0.81 ZAP70 (0.39) SLC7A11ZAP70SRCGHSRMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805816-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2004-07-28 EP disclosed
US-6350767-B1 GROWTH HORMONE RELEASE STIMULANT NOVO NORDISK A/S (DK) 2002-02-26 US disclosed
US-6013658-A ANIMAL GROWTH REGULATORS NOVO NORDISK A/S (DK) 2000-01-11 US disclosed
EP-0907374-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1999-04-14 EP disclosed
WO-1997046252-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1997-12-11 WO disclosed
WO-1996022997-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1996-08-01 WO disclosed