SCHEMBL6603939

SCHEMBL6603939

Cc1nc(C(=O)O)cc2c(NC(=O)NCc3ccc(Cl)cc3Cl)cccc12

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.59
PKM P14618 1/20 0.48
CD38 P28907 1/20 0.45
ROCK2 O75116 2/20 0.45
ROCK1 Q13464 2/20 0.45
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.43
TSHR P16473 1/20 0.43
IDH1 O75874 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GRIK1 P39086 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GSK3B P49841 1/20 0.42
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025727 0.83 TRPV1 (0.66) TRPV1PKMROCK2ROCK1ALDH1A1
SCHEMBL4023559 0.78 TRPV1 (0.67) TRPV1PKMCD38ROCK2ROCK1
SCHEMBL4021114 0.77 TRPV1 (0.63) TRPV1PKMROCK2ROCK1TSHR
SCHEMBL6441785 0.76 TRPV1 (0.60) TRPV1PKMROCK2ROCK1TSHR
SCHEMBL2727166 0.73 TRPV1 (0.61) TRPV1P2RX7
SCHEMBL6066195 0.73 TRPV1 (0.61) TRPV1PKMCD38ROCK2ROCK1
SCHEMBL1932253 0.70 NPC1 (0.64) TRPV1ROCK2ROCK1ALDH1A1IDH1
SCHEMBL6441790 0.69 TSHR (0.45) TRPV1PKMALDH1A1TSHRP2RX7
SCHEMBL6066217 0.69 TRPV1 (0.58) TRPV1P2RX7
SCHEMBL697972 0.68 ALDH1A1 (0.63) ALDH1A1TSHRNPC1RAB9AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478363-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR Abbott Laboratories (US) 2004-11-24 EP disclosed
WO-2003070247-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2003-08-28 WO disclosed