SCHEMBL6604571

SCHEMBL6604571

O=C(O)CCC(=O)c1ccccc1.[NaH]

nearest known ligand 0.95

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.95
ALDH1A1 P00352 5/20 0.83
GAA P10253 1/20 0.83
CYP2C19 P33261 1/20 0.83
LMNA P02545 3/20 0.73
SMN1; SMN2 Q16637 2/20 0.73
RAB9A P51151 2/20 0.73
HIF1A Q16665 2/20 0.73
FFAR1 O14842 1/20 0.73
CYP1A2 P05177 1/20 0.73
HDAC3 O15379 1/20 0.69
HDAC4 P56524 1/20 0.69
HDAC1 Q13547 1/20 0.69
HDAC7 Q8WUI4 1/20 0.69
HDAC2 Q92769 1/20 0.69
HDAC10 Q969S8 1/20 0.69
HDAC11 Q96DB2 1/20 0.69
HDAC8 Q9BY41 1/20 0.69
HDAC6 Q9UBN7 1/20 0.69
HDAC9 Q9UKV0 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL354105 0.98 NR4A2 (1.00) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL7408024 0.95 NR4A2 (0.95) NR4A2ALDH1A1GAACYP2C19LMNA
Water SCHEMBL9863145 0.95 NR4A2 (0.95) NR4A2ALDH1A1GAACYP2C19LMNA
Hydrochloric Acid SCHEMBL1372562 0.95 NR4A2 (0.95) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL6547078 0.95 NR4A2 (0.95) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL1829362 0.91 ALDH1A1 (1.00) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL719034 0.90 NR4A2 (0.85) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL30121738 0.90 NR4A2 (0.85) NR4A2ALDH1A1GAACYP2C19LMNA
SCHEMBL10353454 0.87 NR4A2 (0.81) NR4A2ALDH1A1GAACYP2C19LMNA
Levulinic Acid SCHEMBL4826758 0.87 NR4A2 (0.80) NR4A2ALDH1A1GAACYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142887-B1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE DAVIS & CO (US) 2004-04-07 EP disclosed
EP-0729463-B1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2002-05-22 EP disclosed
EP-1142887-A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE, DAVIS & COMPANY (US) 2001-10-10 EP disclosed
US-5936128-A BENZENETHIOL COMPOUNDS AS INTERMEDIATES; BACTERICIDES, VIRICIDES; HIV WARNER-LAMBERT COMPANY (US) 1999-08-10 US disclosed
US-5840751-A ADMINISTERING IN THE TREATMENT OF INFECTION OR DISEASE CAUSED BY A RETROVIRUS WARNER-LAMBERT COMPANY (US) 1998-11-24 US disclosed
US-5789440-A 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents WARNER-LAMBERT COMPANY (US) 1998-08-04 US disclosed
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729463-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014012-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed