SCHEMBL66046

SCHEMBL66046

Nc1ncnc2c1ncn2[C@H]1C[C@H](O)[C@@H](C(O)Cl)O1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHCY P23526 7/20 0.57
ADA P00813 1/20 0.53
STING1 Q86WV6 1/20 0.53
POLB P06746 1/20 0.52
TP53 P04637 1/20 0.52
CYP2C9 P11712 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
APEX1 P27695 1/20 0.52
PI4KA P42356 1/20 0.52
BLM P54132 1/20 0.52
KMT2A Q03164 1/20 0.52
ADCY1 Q08828 1/20 0.52
PI4K2B Q8TCG2 1/20 0.52
PI4K2A Q9BTU6 1/20 0.52
PI4KB Q9UBF8 1/20 0.52
ENPP1 P22413 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28121858 0.92 AHCY (0.56) AHCYADASTING1POLBTP53
SCHEMBL9875644 0.92 AHCY (0.56) AHCYADASTING1POLBTP53
SCHEMBL4451661 0.92 AHCY (0.59) AHCYADASTING1POLBTP53
SCHEMBL9875640 0.92 AHCY (0.56) AHCYADASTING1POLBTP53
SCHEMBL29375190 0.91 AHCY (0.55) AHCYADASTING1POLBTP53
SCHEMBL2505364 0.91 AHCY (0.55) AHCYADASTING1POLBTP53
SCHEMBL28939795 0.91 AHCY (0.55) AHCYADASTING1POLBTP53
SCHEMBL29739820 0.91 AHCY (0.55) AHCYADASTING1POLBTP53
SCHEMBL30358148 0.90 AHCY (0.52) AHCYADASTING1POLBTP53
SCHEMBL7192503 0.90 AHCY (0.52) AHCYADASTING1POLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2117 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4711364-A1 FUSED PYRROLE RING OR FUSED PYRIDINE RING COMPOUND Pharmaengine, Inc. (TW) 2026-03-18 EP claimed
EP-4701737-A2 MTA-COOPERATIVE PRMT5 INHIBITOR Pharmaengine, Inc. (TW) 2026-03-04 EP claimed
WO-2025077721-A1 MYT1 INHIBITOR BASED ON FUSED THIAZOLE OR PYRIDINE RING PHARMAENGINE, INC. (CN) 2025-04-17 WO claimed
CN-119798282-A Fused pyridine ring-based Myt1 inhibitors 智擎生技制药股份有限公司 2025-04-11 CN claimed
WO-2024222914-A2 MTA-COOPERATIVE PRMT5 INHIBITOR PHARMAENGINE, INC. (CN) 2024-10-31 WO claimed
WO-2023130012-A1 COMPOUNDS FOR MUTANT KRAS PROTEIN DEGRADATION AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2023-07-06 WO claimed
EP-3544685-B1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEV CT BIOTECHNOLOGY (TW) 2023-01-04 EP claimed
EP-3411036-B1 3,5-DISUBSTITUTED PYRAZOLES USEFUL AS CHECKPOINT KINASE 1 (CHK1) INHIBITORS, AND THEIR PREPARATIONS AND APPLICATIONS PHARMAENGINE INC (TW) 2021-12-29 EP claimed
EP-3925625-A1 HYDROPHOBIC MOLECULE-INDUCED BRANCHED POLYMER AGGREGATES AND THEIR USE ANP Technologies, Inc. (US) 2021-12-22 EP claimed
WO-2021222138-A1 COMPOUNDS FOR MUTANT RAS PROTEIN DEGRADATION DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2021-11-04 WO claimed
US-20040241717-A1 Oligomeric compounds for the modulation of thioredoxin expression SANTARIS PHARMA A/S 2004-12-02 US claimed
WO-2004083430-A2 SHORT INTERFERING RNA (siRNA) ANALOGUES SANTARIS PHARMA A/S (DK) 2004-09-30 WO claimed
WO-2004069992-A2 OLIGOMERIC COMPOUNDS FOR THE MODULATION OF RAS EXPRESSION SANTARIS PHARMA A/S (DK) 2004-08-19 WO claimed
WO-2004069991-A2 OLIGOMERIC COMPOUNDS FOR THE MODULATION OF SURVIVIN EXPRESSION SANTARIS PHARMA A/S (DK) 2004-08-19 WO claimed
WO-2004069990-A2 OLIGOMERIC COMPOUNDS FOR THE MODULATION OF THIOREDOXIN EXPRESSION SANTARIS PHARMA A/S (DK) 2004-08-19 WO claimed
US-20040138140-A1 Combination cancer therapy with a GST-activated anticancer compound and another anticancer therapy TELIK, INC. 2004-07-15 US claimed
WO-2004045593-A2 COMBINATION CANCER THERAPY WITH A GST-ACTIVATED ANTICANCER COMPOUND AND ANOTHER ANTICANCER THERAPY TELIK, INC. (US) 2004-06-03 WO claimed
WO-2004020468-A2 INTERFERON BETA-LIKE MOLECULES FOR TREATMENT OF CANCER MAXYGEN APS (DK) 2004-03-11 WO claimed
WO-2003061703-A9 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS WITH STATINS NOVIMMUNE SA (CH) 2003-12-24 WO claimed
WO-1996005865-A1 COMBINATION IMMUNOTOXIN/ANTINEOPLASTIC AGENT THERAPY FOR B-LINEAGE CANCER REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1996-02-29 WO claimed