SCHEMBL6604871

SCHEMBL6604871

O=C(Nc1ccc(Cl)cc1)c1cncs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 1.00
LMNA P02545 4/20 0.58
HTT P42858 1/20 0.58
GRM4 Q14833 1/20 0.56
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
NAMPT P43490 2/20 0.54
MAPK1 P28482 1/20 0.53
GRM5 P41594 1/20 0.49
MAPT P10636 2/20 0.49
NT5E P21589 1/20 0.49
ABL1 P00519 1/20 0.48
MEN1 O00255 2/20 0.48
KDM4E B2RXH2 2/20 0.47
POLB P06746 1/20 0.47
PPARG P37231 1/20 0.47
NR2E3 Q9Y5X4 1/20 0.47
NCOR2 Q9Y618 1/20 0.47
ESR1 P03372 1/20 0.47
ESRRG P62508 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL892318 0.84 KMT2A (0.72) KMT2ALMNAGRM4NPC1RAB9A
SCHEMBL892780 0.83 KMT2A (0.71) KMT2ALMNAHTTGRM4NPC1
SCHEMBL30909377 0.77 KMT2A (0.62) KMT2ALMNAHTTGRM4NPC1
SCHEMBL15886292 0.77 KMT2A (0.72) KMT2ALMNAHTTGRM4NPC1
Ammonia Solution, Strong SCHEMBL20302197 0.75 GRM4 (0.60) KMT2AGRM4NPC1RAB9AMAPK1
SCHEMBL3513684 0.73 TYK2 (0.66)
SCHEMBL7919011 0.73 GRM4 (0.61) KMT2ALMNAGRM4NPC1RAB9A
SCHEMBL11848283 0.73 KMT2A (0.56) KMT2ALMNAGRM4NPC1RAB9A
SCHEMBL10659791 0.73 KMT2A (0.57) KMT2ALMNAGRM4NPC1RAB9A
SCHEMBL3425315 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102535-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-09-29 EP disclosed
EP-1102535-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-05-30 EP disclosed
WO-2000006085-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed