SCHEMBL6605467

SCHEMBL6605467

COc1ccc(N)cc1N(C(C)C)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 3/20 0.46
USP2 O75604 1/20 0.46
CYP19A1 P11511 5/20 0.44
MAPT P10636 3/20 0.44
GAA P10253 3/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 2/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
NQO2 P16083 1/20 0.43
NR4A1 P22736 1/20 0.43
LCK P06239 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
KRAS P01116 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1640545 0.80 APP (0.56) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL1413112 0.76 GAA (0.51) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL18147051 0.75 ALDH1A1 (0.51) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL11338264 0.75 ALDH1A1 (0.47) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL7806591 0.75 GAA (0.44) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL9398336 0.74 MAPT (0.50) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL15486485 0.74 ALDH1A1 (0.46) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL21672910 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EUSP2CYP19A1MAPT
Hydrochloric Acid SCHEMBL15486483 0.73 ALDH1A1 (0.45) ALDH1A1KDM4EUSP2CYP19A1MAPT
SCHEMBL2119806 0.73 ALDH1A1 (0.49) ALDH1A1KDM4ECYP19A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102535-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-09-29 EP disclosed
US-6399656-B1 USING A BENZOPYRAN-3-CARBOXAMIDE COMPOUND SMITHKLINE BEECHAM CORPORATION 2002-06-04 US disclosed
EP-1102535-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-05-30 EP disclosed
WO-2000006085-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed