SCHEMBL6605590

SCHEMBL6605590

CCCCCC1(CCCCC)CC(O)=C(SCc2ccccc2)C(=O)O1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.38
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
MMP13 P45452 2/20 0.38
PRKCA P17252 10/20 0.37
CTSB P07858 1/20 0.36
LDHA P00338 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DAO P14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603220 0.85 LDHA (0.46) S100A4MMP2MMP9MMP8MMP13
SCHEMBL6604705 0.84 LDHA (0.45) S100A4MMP2MMP9MMP8MMP13
SCHEMBL6604082 0.81 LDHA (0.47) S100A4CTSBLDHAKMT2AL3MBTL1
SCHEMBL6603774 0.78 LDHA (0.48) S100A4LDHAKMT2AL3MBTL1DAO
SCHEMBL6606575 0.78 LDHA (0.41) S100A4MMP2MMP9CTSBLDHA
SCHEMBL6604912 0.74 LDHA (0.45) MMP2MMP9MMP8MMP13PRKCA
SCHEMBL6604202 0.74 LDHA (0.59) S100A4LDHADAO
SCHEMBL6603852 0.74 LDHA (0.44) MMP2MMP9MMP8MMP13PRKCA
SCHEMBL6606612 0.72 LDHA (0.49) S100A4LDHAL3MBTL1DAO
SCHEMBL6607615 0.71 LDHA (0.44) S100A4MMP9LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142887-B1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE DAVIS & CO (US) 2004-04-07 EP disclosed
EP-0729463-B1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2002-05-22 EP disclosed
EP-1142887-A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE, DAVIS & COMPANY (US) 2001-10-10 EP disclosed
US-5936128-A BENZENETHIOL COMPOUNDS AS INTERMEDIATES; BACTERICIDES, VIRICIDES; HIV WARNER-LAMBERT COMPANY (US) 1999-08-10 US disclosed
US-5840751-A ADMINISTERING IN THE TREATMENT OF INFECTION OR DISEASE CAUSED BY A RETROVIRUS WARNER-LAMBERT COMPANY (US) 1998-11-24 US disclosed
EP-0729463-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014012-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed