SCHEMBL6605909

SCHEMBL6605909

Nc1ncc(Br)cc1C(=O)Nc1cnccc1CN1CCCC1.Nc1ncc(Br)cc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 2/20 0.47
CCNE1 P24864 2/20 0.47
CDK2 P24941 2/20 0.47
GSK3B P49841 2/20 0.47
TBK1 Q9UHD2 13/20 0.47
IKBKE Q14164 12/20 0.47
PIM2 Q9P1W9 2/20 0.40
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
ATR Q13535 1/20 0.40
PRKCI P41743 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6033879 0.96 TBK1 (0.50) CCNE2CCNE1CDK2GSK3BTBK1
SCHEMBL6035019 0.79 GSK3B (0.61) CCNE2CCNE1CDK2GSK3BTBK1
SCHEMBL6035809 0.74 CACNA1B (0.46) CCNE2CCNE1CDK2GSK3BTBK1
SCHEMBL6033839 0.74 GSK3B (0.74) CCNE2CCNE1CDK2GSK3BTBK1
Hydrochloric Acid SCHEMBL6036000 0.73 GSK3B (0.73) CCNE2CCNE1CDK2GSK3BTBK1
SCHEMBL14059578 0.72 TBK1 (0.58) TBK1IKBKEATRPRKCI
SCHEMBL14059044 0.72 IKBKE (0.55) TBK1IKBKEPRKCI
SCHEMBL6034173 0.70 GSK3B (0.53) CCNE2CCNE1CDK2GSK3BTBK1
SCHEMBL14059394 0.70 PRKCI (0.66) TBK1IKBKEPRKCIGAA
SCHEMBL3146262 0.69 PHF13 (0.50) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP disclosed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO disclosed