SCHEMBL6606097

SCHEMBL6606097

CSc1nccc(Nc2ccc3[nH]ncc3c2)n1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.67
KDR P35968 7/20 0.61
ROCK2 O75116 11/20 0.57
ROCK1 Q13464 4/20 0.57
IGF1R P08069 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26715276 0.83 MAPKAPK2 (0.71) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL3459554 0.80 MAPKAPK2 (0.71) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL20783989 0.80 MAPKAPK2 (1.00) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL26717703 0.80 MAPKAPK2 (0.67) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL18114560 0.76 ROCK2 (0.71) MAPKAPK2KDRROCK2ROCK1
SCHEMBL3810286 0.76 MAPKAPK2 (0.65) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL4879499 0.75 KDR (0.71) MAPKAPK2KDRROCK2ROCK1IGF1R
SCHEMBL18114550 0.75 ROCK2 (0.61) MAPKAPK2KDRROCK2ROCK1
SCHEMBL18792311 0.75 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL18114563 0.74 KDR (0.66) MAPKAPK2KDRROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235806-A4 NOVEL 5-PYRIMIDINECARBOXAMIDE DERIVATIVES AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES DONG WHA PHARM IND CO LTD (KR) 2004-02-04 EP disclosed
EP-1235806-A1 NOVEL 5-PYRIMIDINECARBOXAMIDE DERIVATIVES AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES DONG WHA PHARMACEUTICAL INDUSTRIAL CO. LTD. (KR) 2002-09-04 EP disclosed
WO-2001038308-A1 NOVEL 5-PYRIMIDINECARBOXAMIDE DERIVATIVES AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES DONG WHA PHARM. IND. CO., LTD (KR) 2001-05-31 WO disclosed