SCHEMBL6606402

SCHEMBL6606402

CCC(CCC#CCc1ccc2c(c1)N(C(=O)OC(C)(C)C)CCC2(C)C)c1ccc(C(=O)O)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RARB P10826 7/20 0.39
RARG P13631 7/20 0.39
RARA P10276 6/20 0.39
RXRA P19793 10/20 0.35
RXRB P28702 6/20 0.35
RXRG P48443 4/20 0.35
CYP26A1 O43174 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP26B1 Q9NR63 1/20 0.35
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM1A O60341 1/20 0.33
CRABP2 P29373 1/20 0.33
GPR119 Q8TDV5 1/20 0.32
HNF4A P41235 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6608438 0.92 HDAC1 (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6605497 0.81 KDM1A (0.40) RARBRARGRARAHDAC1HDAC6
SCHEMBL4843508 0.76 RARB (0.47) RARBRARGRARARXRARXRB
SCHEMBL11924574 0.75 KDM1A (0.46) RARBRARARXRARXRBRXRG
SCHEMBL4848988 0.70 KDM1A (0.40) RARBRARGRXRAHDAC1HDAC6
SCHEMBL25515740 0.70 KDM1A (0.49) RARBRARGRARARXRARXRB
SCHEMBL4844192 0.69 KDM1A (0.39) RARBRARGRARARXRAKDM1A
SCHEMBL4847633 0.68 HDAC1 (0.39) RARBRARGRARACYP26A1CYP3A4
SCHEMBL15074679 0.68 KDM1A (0.48) RARBRARGRARACYP3A4HDAC1
SCHEMBL4848678 0.68 KDM1A (0.40) RARBRARGRXRAHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1442032-A1 HETEROCYCLIC RETINOID COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-04 EP disclosed
WO-2003037882-A1 HETEROCYCLIC RETINOID COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2003-05-08 WO disclosed