SCHEMBL6608438

SCHEMBL6608438

CCC(CCC#CCc1ccc2c(c1)N(C(=O)OC(C)(C)C)CCC2(C)C)c1ccc(C(=O)OC)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
PKM P14618 1/20 0.33
CYP3A4 P08684 3/20 0.33
KDM1A O60341 1/20 0.32
KDM4D Q6B0I6 1/20 0.32
RARA P10276 3/20 0.31
RARB P10826 3/20 0.31
CYP26A1 O43174 2/20 0.31
RARG P13631 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606402 0.92 RARB (0.39) HDAC1HDAC6CYP3A4KDM1ARARA
SCHEMBL6605497 0.80 KDM1A (0.40) HDAC1HDAC6KDM1ARARARARB
SCHEMBL4847633 0.76 HDAC1 (0.39) HDAC1HDAC6PKMCYP3A4KDM1A
SCHEMBL11924574 0.76 KDM1A (0.46) HDAC1HDAC6KDM1ARARARARB
SCHEMBL4853701 0.73 HDAC1 (0.39) HDAC1HDAC6PKMCYP3A4KDM1A
SCHEMBL4853714 0.73 HDAC1 (0.39) HDAC1HDAC6PKMCYP3A4KDM1A
SCHEMBL4853709 0.73 HDAC1 (0.39) HDAC1HDAC6PKMCYP3A4KDM1A
SCHEMBL4848988 0.69 KDM1A (0.40) HDAC1HDAC6KDM1ARARBRARG
SCHEMBL4843508 0.68 RARB (0.47) CYP3A4KDM1ARARARARBCYP26A1
SCHEMBL4844192 0.68 KDM1A (0.39) KDM1ARARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1442032-A1 HETEROCYCLIC RETINOID COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-04 EP disclosed
WO-2003037882-A1 HETEROCYCLIC RETINOID COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2003-05-08 WO disclosed