SCHEMBL6606980

SCHEMBL6606980

Cc1cc(COc2ccc(C(=O)[AsH]C3(CC(=O)NO)CCN(C[C@H]4CCCN4C(=O)O)CC3)cc2)c2ccccc2n1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 19/20 0.57
MMP13 P45452 1/20 0.56
ADAMTS4 O75173 2/20 0.52
MMP3 P08254 2/20 0.52
MMP7 P09237 2/20 0.52
ADAMTS1 Q9UHI8 2/20 0.52
ADAMTS5 Q9UNA0 2/20 0.52
MMP8 P22894 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597679 0.88 ADAM17 (0.75) ADAM17MMP13ADAMTS4MMP3MMP7
SCHEMBL6598893 0.80 ADAM17 (0.76) ADAM17MMP13
SCHEMBL6594529 0.78 ADAM17 (0.58) ADAM17
SCHEMBL6596696 0.76 ADAM17 (0.83) ADAM17MMP13ADAMTS4MMP3MMP7
SCHEMBL6598016 0.76 ADAM17 (0.80) ADAM17MMP13ADAMTS4MMP3MMP7
SCHEMBL6598436 0.76 ADAM17 (0.56) ADAM17
SCHEMBL6596146 0.74 ADAM17 (0.78) ADAM17MMP13ADAMTS4MMP3MMP7
SCHEMBL6595238 0.73 ADAM17 (0.56) ADAM17
SCHEMBL6365154 0.73 SPHK2 (0.59) ADAM17
SCHEMBL6595241 0.73 ADAM17 (0.85) ADAM17MMP13ADAMTS4MMP3MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-B1 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL MYERS SQUIBB PHARMA CO (US) 2004-02-25 EP claimed