SCHEMBL6607233

SCHEMBL6607233

CCCC[C@H](NC(=O)O)C(=O)C(=O)Nc1ccccn1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.71
ALOX12 P18054 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.51
HTT P42858 2/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
PKM P14618 2/20 0.50
CTSV O60911 1/20 0.49
CTSS P25774 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
EHMT2 Q96KQ7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604125 1.00 CTSK (0.71) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL5637491 0.78 CTSK (0.53) CTSK
SCHEMBL5637506 0.78 CTSK (0.53) CTSK
SCHEMBL6616469 0.77 HTT (0.50) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL6406963 0.77 HTT (0.50) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL6402731 0.77 HTT (0.50) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL6402737 0.77 HTT (0.50) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL6406973 0.77 HTT (0.50) CTSKALOX12SMN1; SMN2HTTNPC1
SCHEMBL6606767 0.77 CTSK (0.71) CTSKSMN1; SMN2HTTPKMCTSV
SCHEMBL6606757 0.77 CTSK (0.71) CTSKSMN1; SMN2HTTPKMCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1411933-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN K INHIBITORS SmithKline Beecham Corporation (US) 2004-04-28 EP claimed
WO-2003013518-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN K INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-02-20 WO claimed