SCHEMBL6607371

SCHEMBL6607371

Cc1noc(C)c1S(=O)(=O)N(C(=O)[CH]CC(C)C(N)=O)[C@H]1CCCNCC1=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 3/20 0.32
POLB P06746 2/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770196 0.82
SCHEMBL4768440 0.82
SCHEMBL6607376 0.81 TSHR (0.34) TSHRMEN1KMT2AALDH1A1NPSR1
SCHEMBL6589457 0.81
SCHEMBL4761958 0.80 PSEN1 (0.31) MEN1KMT2AALDH1A1
SCHEMBL6602697 0.79 CTSK (0.36)
SCHEMBL6591381 0.79 PSEN1 (0.34)
SCHEMBL6240344 0.79
SCHEMBL6594103 0.79
SCHEMBL4763246 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed