SCHEMBL6607917

SCHEMBL6607917

CCCNc1ccc2[nH]cc(C=O)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
AR P10275 2/20 0.47
CYP2A6 P11509 2/20 0.45
IMPDH2 P12268 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
MPO P05164 5/20 0.43
HTR1D P28221 3/20 0.41
HTR1B P28222 1/20 0.40
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39
HASPIN Q8TF76 1/20 0.39
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2539100 0.78 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL18311437 0.75 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL5403384 0.74 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL11692889 0.74 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19ARCYP2A6
SCHEMBL29935857 0.72 CAPN1 (0.59) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL208051 0.72 CAPN1 (0.59) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL1094048 0.72 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL8257892 0.71 CYP1A2 (0.67) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL29954011 0.71 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL5402406 0.71 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379239-A2 N-(2-ARYLETHYL) BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2004-01-14 EP disclosed
WO-2002078693-A2 N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2002-10-10 WO disclosed