SCHEMBL6609333

SCHEMBL6609333

CC(C)(C)OC(=O)CC[C@@H](CO)NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.45
KMT2A Q03164 2/20 0.44
MDM2 Q00987 1/20 0.44
MDM4 O15151 1/20 0.42
TP53 P04637 1/20 0.42
BACE1 P56817 1/20 0.42
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29687297 1.00 CASP3 (0.45) CASP3KMT2AMDM2MDM4TP53
SCHEMBL29398965 1.00 CASP3 (0.45) CASP3KMT2AMDM2MDM4TP53
SCHEMBL25530715 1.00 CASP3 (0.45) CASP3KMT2AMDM2MDM4TP53
SCHEMBL25530710 0.91 CASP3 (0.44) CASP3KMT2AMDM2MDM4TP53
SCHEMBL16061957 0.91 KMT2A (0.50) CASP3KMT2AMDM2MDM4TP53
SCHEMBL23042740 0.91 CASP3 (0.44) CASP3KMT2AMDM2MDM4TP53
SCHEMBL29687418 0.91 CASP3 (0.44) CASP3KMT2AMDM2MDM4TP53
SCHEMBL29687298 0.91 CASP3 (0.44) CASP3KMT2AMDM2MDM4TP53
SCHEMBL14265315 0.90 CASP3 (0.52) CASP3KMT2AMDM2MDM4TP53
SCHEMBL29400810 0.90 CASP3 (0.52) CASP3KMT2AMDM2MDM4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212309-B1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2004-08-18 EP disclosed
US-6747050-B1 INHIBITING THE ACTIVITY OF CASPASES, PREVENTING INFLAMMATION AND APOPTOSIS LG CHEM INVESTMENT LTD. (KR) 2004-06-08 US disclosed
EP-1212309-A4 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2002-11-27 EP disclosed
EP-1212309-A1 CASPASE INHIBITOR LG Chem Investment, Ltd. (KR) 2002-06-12 EP disclosed
WO-2001021600-A1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD. (KR) 2001-03-29 WO disclosed
WO-2001021599-A1 CASPASE INHIBITOR LG CHEMICAL LTD. (KR) 2001-03-29 WO disclosed