SCHEMBL6609781

SCHEMBL6609781

CN(C)c1ccc(N2CC(OC(=O)O)CC2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MAPT P10636 4/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MCL1 Q07820 1/20 0.46
HIF1A Q16665 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GAA P10253 3/20 0.41
TSHR P16473 3/20 0.39
MAPK1 P28482 2/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
CA6 P23280 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
CA5B Q9Y2D0 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6614023 0.85 TSHR (0.55) ALDH1A1MAPTHPGDSMN1; SMN2TSHR
SCHEMBL6613573 0.83 POLB (0.49) ALDH1A1MAPTHPGDSMN1; SMN2TSHR
SCHEMBL2766821 0.82 RXFP1 (0.52) ALDH1A1MAPTSMN1; SMN2MAPK1CA12
SCHEMBL6613333 0.81 TP53 (0.48) MAPTHPGDSMN1; SMN2TSHRMAPK1
SCHEMBL6609944 0.81 MAPT (0.49) ALDH1A1MAPTHPGDSMN1; SMN2KDM4E
SCHEMBL5844388 0.79 CA12 (0.60) ALDH1A1MAPTHPGDSMN1; SMN2KDM4E
SCHEMBL5739319 0.78 ALDH1A1 (0.56) ALDH1A1MAPTHPGDSMN1; SMN2TSHR
SCHEMBL6206173 0.78 MCHR1 (0.43) MAPTTP53
SCHEMBL5735257 0.77 MAPT (0.55) ALDH1A1MAPTSMN1; SMN2KDM4EGAA
SCHEMBL6610780 0.75 MAPT (0.53) ALDH1A1MAPTHPGDNPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463724-A1 PYRROLIDONE CARBOXAMIDES Actelion Pharmaceuticals Ltd. (CH) 2004-10-06 EP disclosed
WO-2003059905-A1 PYRROLIDONE CARBOXAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2003-07-24 WO disclosed