SCHEMBL6609968

SCHEMBL6609968

O=C(Nc1c[c]ccc1)N1CCCC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
NPSR1 Q6W5P4 2/20 0.55
RECQL P46063 1/20 0.55
RAB9A P51151 6/20 0.54
TSHR P16473 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
NPC1 O15118 4/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 1/20 0.51
TGM2 P21980 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL962960 0.86 CYP2C9 (0.68) ALDH1A1KMT2AMEN1NPSR1RAB9A
SCHEMBL27472376 0.80 TRPV1 (0.62) ALDH1A1KMT2AMEN1TSHRCA12
SCHEMBL751780 0.80 RAB9A (0.62) ALDH1A1KMT2AMEN1NPSR1RECQL
SCHEMBL4776281 0.79 CYP2C9 (0.71) ALDH1A1KMT2AMEN1NPSR1RECQL
SCHEMBL754698 0.78 RAB9A (0.65) ALDH1A1KMT2AMEN1NPSR1RAB9A
Hydrochloric Acid SCHEMBL7128759 0.78 POLB (0.72) ALDH1A1KMT2AMEN1NPSR1RECQL
SCHEMBL420582 0.78 RAB9A (0.69) ALDH1A1KMT2AMEN1NPSR1RECQL
SCHEMBL4051171 0.78 RAB9A (0.69) ALDH1A1KMT2AMEN1NPSR1RECQL
SCHEMBL751658 0.76 RAB9A (0.57) ALDH1A1KMT2AMEN1NPSR1RAB9A
SCHEMBL4901874 0.76 POLB (0.67) ALDH1A1KMT2AMEN1RECQLRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140895-B1 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO (JP) 2004-03-24 EP claimed
WO-2003018019-A2 NEW USE OF CYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-03-06 WO claimed
CN-1343206-A Cyclocompound FUJISAWA PHARMACEUTICAL CO (JP) 2002-04-03 CN claimed
EP-1140895-A2 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP claimed
WO-2000040576-A2 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-13 WO claimed
EP-1140895-B1 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO (JP) 2004-03-24 EP disclosed
CN-1343206-A Cyclocompound FUJISAWA PHARMACEUTICAL CO (JP) 2002-04-03 CN disclosed
EP-1140895-A2 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP disclosed
WO-2000040576-A2 THIOPYRAN COMPOUNDS AS INHIBITORS OF MMP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-13 WO disclosed