SCHEMBL661435

SCHEMBL661435

COc1cc(I)c(C(C)=O)cc1OC(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
CYP3A4 P08684 1/20 0.43
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
ACHE P22303 1/20 0.39
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
BRPF1 P55201 1/20 0.37
LMNA P02545 1/20 0.37
IRAK4 Q9NWZ3 2/20 0.37
HMGCR P04035 1/20 0.37
PDE4B Q07343 2/20 0.36
PDE4A P27815 2/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL661287 0.84 HMGCR (0.54) HTTCYP3A4LCKFYNACHE
SCHEMBL660608 0.83 LCK (0.59) HTTCYP3A4LCKFYNACHE
SCHEMBL31081166 0.83 LCK (0.59) HTTCYP3A4LCKFYNACHE
SCHEMBL10101864 0.81 IRAK4 (0.38) HTTCYP3A4BRPF1IRAK4ALDH1A1
SCHEMBL14042389 0.80 HTT (0.51) HTTCYP3A4LCKFYNACHE
SCHEMBL660858 0.77 HTT (0.56) HTTCYP3A4RAB9AKDM4ELMNA
SCHEMBL22595755 0.77 HTT (0.47) HTTCYP3A4LCKFYNRAB9A
SCHEMBL28786056 0.75 LCK (0.77) HTTLCKFYNKDM4EALDH1A1
SCHEMBL18312021 0.75 LCK (0.56) HTTCYP3A4LCKFYNKDM4E
SCHEMBL661243 0.75 MGAM (0.42) CYP3A4ACHELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8536157-B2 Non-steroidal compounds THE UNIVERSITY OF MELBOURNE (AU) 2013-09-17 US disclosed
US-8536157-B2 Non-steroidal compounds THE UNIVERSITY OF MELBOURNE (AU) 2013-09-17 US disclosed
US-20120046255-A1 NON-STEROIDAL COMPOUNDS THE UNIVERSITY OF MELBOURNE of ROYAL PARADE PARKVILLE (AU) 2012-02-23 US disclosed
US-20120046255-A1 NON-STEROIDAL COMPOUNDS THE UNIVERSITY OF MELBOURNE of ROYAL PARADE PARKVILLE (AU) 2012-02-23 US disclosed
WO-2008124878-A1 NON-STEROIDAL COMPOUNDS CRYPTOPHARMA PTY LTD (AU) 2008-10-23 WO disclosed
WO-2008124878-A1 NON-STEROIDAL COMPOUNDS CRYPTOPHARMA PTY LTD (AU) 2008-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046255-A1 NON-STEROIDAL COMPOUNDS PTGES2, PTGES, PTGES3 HTT 3412/4885CYP3A4 500/4885LCK 3485/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.