SCHEMBL6614764

SCHEMBL6614764

NC(=O)C1CC(F)(F)CN1C(=O)CCl

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 15/20 0.40
CNR1 P21554 1/20 0.38
OPRM1 P35372 2/20 0.36
OPRK1 P41145 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1345807 1.00 CNR2 (0.40) CNR2CNR1OPRM1OPRK1MAOA
SCHEMBL1493746 0.85 CNR2 (0.42) CNR2CNR1OPRM1OPRK1RORC
SCHEMBL1493865 0.85 CNR2 (0.42) CNR2CNR1OPRM1OPRK1RORC
SCHEMBL2845977 0.79 CNR2 (0.41) CNR2CNR1OPRM1OPRK1MAOA
SCHEMBL28038908 0.79 CNR2 (0.41) CNR2CNR1OPRM1OPRK1MAOA
SCHEMBL15129890 0.79 CNR2 (0.41) CNR2CNR1OPRM1OPRK1MAOA
SCHEMBL25494519 0.75 OPRM1 (0.42) CNR2CNR1OPRM1OPRK1
SCHEMBL1347339 0.72 DPP4 (0.53)
SCHEMBL15130403 0.71 HDAC8 (0.46) CNR2MAOAMAOB
SCHEMBL29162891 0.71 CNR2 (0.37) CNR2CNR1OPRM1OPRK1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487807-A2 NEW COMPOUNDS Sanofi-Aventis (FR) 2004-12-22 EP disclosed
WO-2003074500-A2 N-AMINOACETYL-PYRROLIDINE-2-CARBONITRILES AND THEIR USE AS DDP-IV INHIBITORS SANOFI-AVENTIS (FR) 2003-09-12 WO disclosed