SCHEMBL6614907

SCHEMBL6614907

COc1ccc(CN2CCC3(CC2)C(=O)NC(CC(C)C)C(=O)N3Cc2ccccn2)cc1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.69
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482157 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6612591 0.91 CCR5 (0.80) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL7534522 0.91 CCR5 (0.71) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6613691 0.90 CCR5 (0.69) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6612792 0.89 CCR5 (0.86) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6614578 0.89 CCR5 (0.86) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6615696 0.87 CCR5 (0.71) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6614881 0.86 CCR5 (0.91) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6613696 0.86 CCR5 (0.78) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6614551 0.85 CCR5 (0.74) CCR5CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed