SCHEMBL6615982

SCHEMBL6615982

CCCN1C(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C12CCN(CCCCCc1ccccc1)CC2

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.69
CXCR4 P61073 2/20 0.63
CXCR3 P49682 1/20 0.56
HTR1A P08908 1/20 0.51
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A4 P31645 1/20 0.51
HRH1 P35367 1/20 0.51
DRD3 P35462 1/20 0.51
HTR2B P41595 1/20 0.51
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613194 1.00 CCR5 (0.69) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6612324 1.00 CCR5 (0.69) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6611712 0.99 CCR5 (0.68) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6613104 0.97 CCR5 (0.65) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6012533 0.94 CCR5 (0.60) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6012467 0.94 CCR5 (0.60) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6613915 0.94 CCR5 (0.60) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6610609 0.93 CCR5 (0.59) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6617863 0.93 CCR5 (0.59) CCR5CXCR4CXCR3HTR1ADRD2
SCHEMBL6012206 0.93 CCR5 (0.59) CCR5CXCR4CXCR3HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed