SCHEMBL6616243

SCHEMBL6616243

CC(C)CONC1=NS(=O)(=O)c2cnccc2N1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6621856 0.87 CA12 (0.33) CA12CA1CA2CA9ALDH1A1
SCHEMBL6616327 0.85 CA12 (0.36) CA12CA1CA2CA9ALDH1A1
SCHEMBL6617236 0.83 CA12 (0.36) CA12CA1CA2CA9ALDH1A1
SCHEMBL8623804 0.82 KDM6B (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL6616356 0.81
SCHEMBL6618067 0.81 NAMPT (0.37) CA12CA1CA2CA9ALDH1A1
SCHEMBL6617764 0.81 HCAR3 (0.38) CA12CA1CA2CA9ALDH1A1
SCHEMBL8626480 0.80 CA12 (0.36) CA12CA1CA2CA9ALDH1A1
SCHEMBL6618114 0.80 UTS2R (0.32) CA12CA1CA2CA9ALDH1A1
SCHEMBL6619415 0.79 TAAR1 (0.37) CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877748-B1 PYRIDO-1,2,4-THIADIAZINE AND PYRIDO-1,4-THIAZINE DERIVATIVES, THEIR PREPARATION AND USE UNIV LIEGE (BE) 2004-11-03 EP disclosed
US-5792764-A ENDOCRINE DISORDERS ESPECIALLY AS A K(ATP)-CHANNEL MODULATOR NOVO NORDISK A/S (DK) 1998-08-11 US disclosed