SCHEMBL6616730

SCHEMBL6616730

CCCN1C(=O)C(CC(C)C)NC(=O)C12CCN(S(=O)(=O)c1ccccc1C(=O)OC)CC2

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.55
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CXCR4 P61073 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6615639 0.84 CCR5 (0.59) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6613731 0.83 CCR5 (0.59) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6613285 0.82 CCR5 (0.47) CCR5
SCHEMBL6613555 0.81 CCR5 (0.58) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6615476 0.79 CCR5 (0.56) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6012502 0.79 CCR5 (0.58) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6611360 0.79 CCR5 (0.58) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6012399 0.78 CCR5 (0.56) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6012384 0.78 CCR5 (0.56) CCR5CYP3A4CYP2D6CYP2C9CXCR4
SCHEMBL6614484 0.78 CCR5 (0.54) CCR5CYP3A4CYP2D6CYP2C9CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed