SCHEMBL6617

SCHEMBL6617

Cc1noc(-c2ccc(Br)cc2)c1CCC/C=C/c1ccc(Cl)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HTT P42858 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
P2RX7 Q99572 1/20 0.33
ALOX15 P16050 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
BRD4 O60885 2/20 0.31
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587 0.80 BRD4 (0.33) HDAC1BRD4GRIK1GRIK2
SCHEMBL13720099 0.80 BRD4 (0.33) HDAC1BRD4GRIK1GRIK2
SCHEMBL10012 0.71 CYP2C9 (0.40) CYP1A2CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL27870816 0.71 CYP1A2 (0.42) HDAC1HTTCYP1A2CYP3A4CYP2C9
SCHEMBL1652 0.70 CYP1A2 (0.41) HDAC1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7129 0.68 BRD4 (0.36) HDAC1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL18597812 0.68 CYP1A2 (0.44) HTTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1185 0.68 CYP1A2 (0.44) HTTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6483 0.67 CYP1A2 (0.43) HTTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1683 0.67 CYP1A2 (0.43) HTTCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed