SCHEMBL6620183

SCHEMBL6620183

Cc1ccccc1-c1cnc(N)c(C(=O)Nc2cccnc2)n1

nearest known ligand 0.81

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 15/20 0.81
PRKDC P78527 4/20 0.81
CYP3A4 P08684 1/20 0.67
GSK3B P49841 4/20 0.64
CCNE2 O96020 3/20 0.64
CCNE1 P24864 3/20 0.64
CDK2 P24941 3/20 0.64
PRKCI P41743 1/20 0.59
ATM Q13315 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2485557 0.90 ATR (1.00) ATRPRKDCCYP3A4ATM
SCHEMBL6616666 0.87 ATR (0.81) ATRPRKDCCYP3A4GSK3BCCNE2
SCHEMBL6615544 0.84 ATR (0.88) ATRPRKDCCYP3A4GSK3BCCNE2
SCHEMBL6035902 0.83 GSK3B (0.69) ATRPRKDCCYP3A4GSK3BCCNE2
SCHEMBL6616728 0.83 ATR (0.67) ATRPRKDCCYP3A4GSK3BCCNE2
SCHEMBL6615738 0.83 CCNE2 (0.68) ATRCYP3A4GSK3BCCNE2CCNE1
SCHEMBL2484903 0.80 ATR (1.00) ATRPRKDCCYP3A4ATM
SCHEMBL6616579 0.80 ATR (0.66) ATRCYP3A4GSK3BCCNE2CCNE1
SCHEMBL6618758 0.80 ATR (0.63) ATRPRKDCCYP3A4GSK3BCCNE2
SCHEMBL6616188 0.80 ATR (0.68) ATRCYP3A4GSK3BCCNE2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040186113-A1 Heterocyclic amines for the treatment of conditions associated with gsk-3 ASTRAZENECA AB (SE) 2004-09-23 US claimed
US-20040186113-A1 Heterocyclic amines for the treatment of conditions associated with gsk-3 ASTRAZENECA AB (SE) 2004-09-23 US disclosed
EP-1406877-A1 HETEROCYCLIC AMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-04-14 EP disclosed
WO-2003004475-A1 HETEROCYCLIC AMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040186113-A1 Heterocyclic amines for the treatment of conditions associated with gsk-3 GSK3A, GSK3B, PYGL ATR 1381/4885PRKDC 897/4885CYP3A4 1187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.