SCHEMBL6622952

SCHEMBL6622952

CCn1c(N)nc2cc(NC)ccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
KDM4E B2RXH2 3/20 0.48
RAD52 P43351 1/20 0.48
TLR8 Q9NR97 4/20 0.47
POLB P06746 2/20 0.43
CNR2 P34972 1/20 0.43
ITK Q08881 1/20 0.42
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NUDT1 P36639 1/20 0.40
BACE1 P56817 1/20 0.40
KMT2A Q03164 1/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NLRP3 Q96P20 1/20 0.39
RPS6KA5 O75582 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201782 0.83 KDM4E (0.60) HTTCYP1A2KDM4ERAD52ALDH1A1
SCHEMBL21310890 0.81 BACE1 (0.39) HTTCYP1A2CYP2D6KDM4ERAD52
SCHEMBL6023581 0.79 ITK (0.59) TLR8ITKNUDT1BACE1
SCHEMBL12598268 0.79 TLR8 (0.70) HTTCYP1A2CYP2D6KDM4ERAD52
SCHEMBL979555 0.78 HTT (0.60) HTTCYP1A2CYP2D6KDM4ERAD52
Dimethylamine SCHEMBL6930952 0.76 CYP1A2 (0.90) HTTCYP1A2CYP2D6KDM4ETLR8
Dimethylamine SCHEMBL6934118 0.74 CYP1A2 (0.87) HTTCYP1A2CYP2D6KDM4ETLR8
SCHEMBL14521693 0.74 CYP1A2 (0.55) HTTCYP1A2CYP2D6KDM4ERAD52
SCHEMBL1992429 0.73 CYP1A2 (1.00) HTTCYP1A2CYP2D6KDM4ETLR8
SCHEMBL18327521 0.73 HTT (0.54) HTTCYP1A2CYP2D6KDM4ERAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-A1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-12-22 EP disclosed
WO-2003074515-A1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-09-12 WO disclosed