SCHEMBL6623237

SCHEMBL6623237

Cc1ccccc1-c1[c]c[nH]n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
PKM P14618 1/20 0.42
NOTUM Q6P988 1/20 0.42
GAA P10253 1/20 0.42
IDO1 P14902 1/20 0.42
METAP2 P50579 1/20 0.42
NPSR1 Q6W5P4 3/20 0.39
DCUN1D1 Q96GG9 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PRNP P04156 1/20 0.39
PPARG P37231 1/20 0.39
MAPK10 P53779 1/20 0.39
NCOA2 Q15596 1/20 0.39
NCOA1 Q15788 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
RAB9A P51151 6/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
NPC1 O15118 5/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292087 0.72 NR1H2 (0.38)
SCHEMBL7853517 0.70 NOTUM (0.45) NOTUMIDO1TSHR
SCHEMBL2764413 0.68 NOTUM (0.39) ALDH1A1NOTUMMETAP2DCUN1D1RAB9A
SCHEMBL3818490 0.65 NPC1 (0.38) ALDH1A1PKMNOTUMGAAIDO1
SCHEMBL28587436 0.65 DCUN1D1 (0.41) ALDH1A1PKMNOTUMGAAIDO1
SCHEMBL197690 0.65 ACHE (0.64) ALDH1A1GAAIDO1METAP2DCUN1D1
SCHEMBL30354037 0.65 ACHE (0.64) ALDH1A1GAAIDO1METAP2DCUN1D1
SCHEMBL30169568 0.65 ACHE (0.64) ALDH1A1GAAIDO1METAP2DCUN1D1
SCHEMBL11620981 0.64 DCUN1D1 (0.44) ALDH1A1PKMNOTUMGAAIDO1
SCHEMBL11624680 0.64 IDO1 (0.53) ALDH1A1PKMNOTUMGAAIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490340-A1 HETEROAROMATIC UREA DERIVATIVES AS VR-1 RECEPTOR MODULATORS FOR TREATING PAIN MERCK SHARP & DOHME LTD. (GB) 2004-12-29 EP disclosed
WO-2003080578-A1 HETEROAROMATIC UREA DERIVATIVES AS VR-1 RECEPTOR MODULATORS FOR TREATING PAIN MERCK SHARP & DOHME LIMITED (GB) 2003-10-02 WO disclosed
EP-1000055-A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS G.D. Searle & Co. (US) 2000-05-17 EP disclosed
WO-1998052940-A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS G.D. SEARLE AND CO. (US) 1998-11-26 WO disclosed