SCHEMBL6623933

SCHEMBL6623933

CC1CN(c2cc(N3CCOCC3)nc(-n3cnc4ccccc43)n2)CC(C)O1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 3/20 0.62
LCK P06239 3/20 0.56
PDCD1 Q15116 6/20 0.51
CD274 Q9NZQ7 6/20 0.51
CHEK1 O14757 4/20 0.51
ATR Q13535 4/20 0.51
ATRIP Q8WXE1 4/20 0.51
HRH4 Q9H3N8 1/20 0.47
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
GAA P10253 2/20 0.46
PIK3CD O00329 1/20 0.46
HPGD P15428 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
MTOR P42345 2/20 0.43
PIK3R1 P27986 1/20 0.43
PIK3CA P42336 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6626217 1.00 PIK3CB (0.62) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6623928 1.00 PIK3CB (0.62) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6626223 1.00 PIK3CB (0.62) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6626337 0.92 KDM4E (0.53) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6626331 0.92 KDM4E (0.53) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6625645 0.89 PIK3CB (0.78) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6628042 0.88 PIK3CB (0.77) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6628039 0.88 PIK3CB (0.77) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6625695 0.88 PIK3CB (0.77) PIK3CBLCKPDCD1CD274CHEK1
SCHEMBL6625690 0.88 PIK3CB (0.77) PIK3CBLCKPDCD1CD274CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020462-B1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KK (JP) 2004-02-11 EP disclosed
US-6251900-B1 Heterocyclic compounds and antitumor agent containing the same as active ingredient ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2001-06-26 US disclosed
EP-1020462-A1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed