SCHEMBL6624906

SCHEMBL6624906

CC1(C)CN(c2cc(N3CCOCC3)nc(-n3cnc4ccccc43)n2)CCO1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 3/20 0.61
LCK P06239 3/20 0.55
HRH4 Q9H3N8 1/20 0.47
PDCD1 Q15116 5/20 0.46
CD274 Q9NZQ7 5/20 0.46
ATR Q13535 5/20 0.46
CHEK1 O14757 4/20 0.46
ATRIP Q8WXE1 4/20 0.46
PIK3CD O00329 1/20 0.43
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
PRKDC P78527 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 1/20 0.41
PIK3CA P42336 1/20 0.40
MAP3K12 Q12852 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6624867 0.88 PIK3CB (0.76) PIK3CBLCKPDCD1CD274ATR
SCHEMBL6625645 0.88 PIK3CB (0.78) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6626031 0.85 PIK3CB (0.74) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6625425 0.84 PIK3CB (0.67) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6626232 0.83 PIK3CB (0.70) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL4118961 0.82 PIK3CB (0.69) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6625181 0.81 PIK3CB (0.67) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6625200 0.81 PIK3CB (0.74) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6624863 0.81 PIK3CB (0.66) PIK3CBLCKHRH4PDCD1CD274
SCHEMBL6623979 0.80 PIK3CB (0.69) PIK3CBLCKHRH4PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020462-B1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KK (JP) 2004-02-11 EP disclosed
US-6251900-B1 Heterocyclic compounds and antitumor agent containing the same as active ingredient ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2001-06-26 US disclosed
EP-1020462-A1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed