SCHEMBL6625425

SCHEMBL6625425

CN1CCN(c2cc(N3CCOCC3)nc(-n3cnc4ccccc43)n2)CC1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 3/20 0.67
HRH4 Q9H3N8 2/20 0.66
LCK P06239 2/20 0.60
NPSR1 Q6W5P4 1/20 0.52
JAK2 O60674 4/20 0.50
JAK3 P52333 4/20 0.50
PDCD1 Q15116 5/20 0.49
CD274 Q9NZQ7 5/20 0.49
CHEK1 O14757 4/20 0.49
ATR Q13535 4/20 0.49
ATRIP Q8WXE1 4/20 0.49
MKNK1 Q9BUB5 2/20 0.49
MKNK2 Q9HBH9 1/20 0.47
PIK3CD O00329 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6625645 0.93 PIK3CB (0.78) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6626031 0.90 PIK3CB (0.74) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6627240 0.89 PIK3CB (0.85) PIK3CBHRH4LCKNPSR1MKNK1
SCHEMBL6626232 0.88 PIK3CB (0.70) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL4118961 0.87 PIK3CB (0.69) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625181 0.86 PIK3CB (0.67) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625200 0.85 PIK3CB (0.74) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6624863 0.85 PIK3CB (0.66) PIK3CBHRH4LCKJAK2JAK3
SCHEMBL6623979 0.85 PIK3CB (0.69) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6626217 0.84 PIK3CB (0.62) PIK3CBHRH4LCKNPSR1PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020462-B1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KK (JP) 2004-02-11 EP disclosed
US-6251900-B1 Heterocyclic compounds and antitumor agent containing the same as active ingredient ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2001-06-26 US disclosed
EP-1020462-A1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed