SCHEMBL6625517

SCHEMBL6625517

O[C@@H]1CN(CCc2ccccc2)CC[C@@H]1c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
LTA4H P09960 4/20 0.56
EPHX2 P34913 2/20 0.52
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
OPRM1 P35372 1/20 0.48
KDM4E B2RXH2 2/20 0.48
GRIN1 Q05586 1/20 0.47
GRIN2B Q13224 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
S1PR5 Q9H228 1/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6625519 1.00 HRH3 (0.57) HRH3NPC1RAB9ALTA4HEPHX2
SCHEMBL11559799 0.87 CCR5 (0.55) OPRM1
SCHEMBL11559798 0.87 CCR5 (0.55) OPRM1
SCHEMBL11559870 0.87 CCR5 (0.55) OPRM1
SCHEMBL11559805 0.87 CCR5 (0.55) OPRM1
SCHEMBL11559861 0.87 CCR5 (0.55) OPRM1
SCHEMBL3069231 0.80 NPC1 (0.52) HRH3NPC1RAB9AKDM4EALDH1A1
SCHEMBL16897870 0.79 NPC1 (0.51) HRH3NPC1RAB9AKDM4EGRIN1
SCHEMBL16897945 0.79 NPC1 (0.51) HRH3NPC1RAB9AKDM4EGRIN1
SCHEMBL6951299 0.78 NPC1 (0.50) HRH3NPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979824-B1 Process for the preparation of substituted piperidine-epoxides HOFFMANN LA ROCHE (CH) 2004-10-06 EP claimed