SCHEMBL6627445

SCHEMBL6627445

O=C(O)CC[C@H](NC(=O)[C@@H]1CCCN2C(=O)CC[C@H](NS(=O)(=O)c3ccc(C(F)(F)F)cc3)C(=O)N12)C(=O)COC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.40
IL1B P01584 2/20 0.39
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
LCK P06239 10/20 0.34
CASP3 P42574 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6670787 0.91 CASP1 (0.36) CASP1IL1BMMEACELCK
SCHEMBL6626820 0.91 CASP1 (0.38) CASP1IL1BMMEACELCK
SCHEMBL6626823 0.91 CASP1 (0.38) CASP1IL1BMMEACELCK
SCHEMBL6629028 0.91 CASP1 (0.40) CASP1IL1BMMEACELCK
SCHEMBL6629031 0.91 CASP1 (0.40) CASP1IL1BMMEACELCK
SCHEMBL6627405 0.88 CASP1 (0.44) CASP1IL1BMMEACELCK
SCHEMBL6626880 0.88 CASP1 (0.38) CASP1IL1BMMEACELCK
SCHEMBL7089222 0.85 CASP1 (0.35) CASP1IL1BMMEACELCK
SCHEMBL6626824 0.84 CASP1 (0.38) CASP1IL1BMMEACELCK
SCHEMBL6631460 0.82 CASP1 (0.48) CASP1IL1BMMEACELCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246824-B1 CARBOXAMIDE DIAZEPIN DERIVATIVES, PREPARATION METHOD, USE AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF AVENTIS PHARMA SA (FR) 2004-06-09 EP claimed
EP-1246824-B1 CARBOXAMIDE DIAZEPIN DERIVATIVES, PREPARATION METHOD, USE AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF AVENTIS PHARMA SA (FR) 2004-06-09 EP disclosed