SCHEMBL6628735

SCHEMBL6628735

COc1cccc(C(=O)NC2CCC(=O)N3CCC[C@@H](C(=O)N[C@@H](Cc4ccccc4)C(=O)COC(=O)c4c(Cl)cccc4Cl)N3C2=O)c1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 4/20 0.50
LCK P06239 15/20 0.49
IL1B P01584 1/20 0.47
MME P08473 1/20 0.45
ACE P12821 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6628733 1.00 CASP1 (0.50) CASP1LCKIL1BMMEACE
SCHEMBL6628994 0.91 CASP1 (0.50) CASP1LCKIL1B
SCHEMBL6626534 0.91 CASP1 (0.50) CASP1LCKIL1B
SCHEMBL6628738 0.87 CASP1 (0.51) CASP1LCKIL1BMMEACE
SCHEMBL6627304 0.86 LCK (0.48) CASP1LCKIL1BMMEACE
SCHEMBL6627306 0.86 LCK (0.48) CASP1LCKIL1BMMEACE
SCHEMBL6629364 0.86 CASP1 (0.50) CASP1LCKIL1BMMEACE
SCHEMBL645039 0.85 CASP1 (0.64) CASP1LCKIL1BMMEACE
SCHEMBL10247734 0.85 CASP1 (0.64) CASP1LCKIL1BMMEACE
SCHEMBL646652 0.85 CASP1 (0.64) CASP1LCKIL1BMMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246824-B1 CARBOXAMIDE DIAZEPIN DERIVATIVES, PREPARATION METHOD, USE AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF AVENTIS PHARMA SA (FR) 2004-06-09 EP claimed