SCHEMBL6630686

SCHEMBL6630686

Cc1ccc(Oc2ccc(C(N)=O)cc2)s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 16/20 0.58
PARP15 Q460N3 4/20 0.58
PARP4 Q9UKK3 2/20 0.58
PARP14 Q460N5 2/20 0.58
ALDH1A1 P00352 1/20 0.58
KMT2A Q03164 1/20 0.58
PARP16 Q8N5Y8 1/20 0.58
PARP11 Q9NR21 1/20 0.58
PARP2 Q9UGN5 3/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
PARP1 P09874 1/20 0.50
PARP3 Q9Y6F1 1/20 0.47
TNKS O95271 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46
F2 P00734 1/20 0.41
PRSS1 P07477 1/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
ST14 Q9Y5Y6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6631259 0.83 PARP10 (0.64) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL6633394 0.80 PARP10 (0.58) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL4964075 0.78 PARP10 (0.57) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL3137816 0.75 PARP10 (1.00) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL24592196 0.74 PARP10 (0.79) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL3013339 0.74 PARP10 (0.79) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL6631091 0.72 PARP10 (0.62) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL5697485 0.72 LTA4H (0.46)
SCHEMBL6630663 0.71 PARP10 (0.79) PARP10PARP15PARP4PARP14ALDH1A1
SCHEMBL25352415 0.71 DAO (0.42) ALDH1A1KMT2ASENP8SENP6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1248787-B1 NOVEL SUBTITUTED PYRAZOLO[4,3-e]DIAZEPINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, USE AS MEDICINAL PRODUCTS AND PROCESSES FOR PREPARING THEM WARNER LAMBERT CO (US) 2004-10-06 EP claimed
EP-1480977-A2 SUBSTITUTED ARYL COMPOUNDS FOR TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-12-01 EP disclosed
WO-2003070728-A2 AZABICYCLO-SUBSTITUTED BENZOYLAMIDES AND THIOAMIDES FOR TREATMENT OF CNS-RELATED DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2003-08-28 WO disclosed