SCHEMBL6631444

SCHEMBL6631444

[N-]=[N+]=CC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H]1CCCN2C(=O)CC[C@H](NC(=O)NC3CCCCC3)C(=O)N12

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.47
IL1B P01584 2/20 0.44
MME P08473 2/20 0.41
ACE P12821 2/20 0.41
LCK P06239 11/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630785 0.88 CASP1 (0.48) CASP1IL1BMMEACELCK
SCHEMBL6630998 0.88 CASP1 (0.44) CASP1IL1BMMEACELCK
SCHEMBL6626944 0.88 CASP1 (0.44) CASP1IL1BMMEACELCK
SCHEMBL6631451 0.86 CASP1 (0.43) CASP1IL1BMMEACELCK
SCHEMBL6628317 0.85 CASP1 (0.42) CASP1IL1BMMEACELCK
SCHEMBL6627788 0.85 CASP1 (0.44) CASP1IL1BMMEACELCK
SCHEMBL6627923 0.85 CASP1 (0.52) CASP1IL1BMMEACELCK
SCHEMBL6627184 0.83 CASP1 (0.48) CASP1IL1BMMEACELCK
SCHEMBL645114 0.81 CASP1 (0.54) CASP1IL1BMMEACELCK
SCHEMBL6627216 0.80 CASP1 (0.54) CASP1IL1BLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246824-B1 CARBOXAMIDE DIAZEPIN DERIVATIVES, PREPARATION METHOD, USE AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF AVENTIS PHARMA SA (FR) 2004-06-09 EP claimed