SCHEMBL6634573

SCHEMBL6634573

COC(=O)[C@H](Cc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1)NC(=O)c1ccc(C(=O)Nc2cccc(O)c2)cc1Cl

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.66
ITGA4 P13612 20/20 0.66
ITGA2 P17301 1/20 0.50
ITGB7 P26010 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874286 0.90 ITGB1 (0.81) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6641695 0.90 ITGB1 (0.80) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6637322 0.84 ITGB1 (0.68) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15147586 0.82 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15147585 0.82 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6663322 0.81 ITGB1 (0.83) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6639689 0.81 ITGB1 (0.62) ITGB1ITGA4ITGA2ITGB7
SCHEMBL27682872 0.80 ITGB1 (0.75) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6642500 0.80 ITGB1 (0.75) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15143334 0.80 ITGB1 (0.51) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005445-B1 N-ALKANOYLPHENYLALANINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-05-26 EP disclosed
EP-1403247-A1 N-Alkanoylphenylalanine derivatives F.HOFFMANN-LA ROCHE AG (CH) 2004-03-31 EP disclosed
US-6229011-B1 BINDING INHIBITORS BETWEEN VASCULAR ADHESION MOLECULE-1 AND ALPHA. BETA.INTEGRIN; USEFUL FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES SUCH AS MULTIPLE SCLEROSIS, ASTHMA, AND INFLAMMATORY BOWEL DISEASE HOFFMAN-LA ROCHE INC. 2001-05-08 US disclosed
EP-1005445-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-07 EP disclosed
WO-1999010312-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-04 WO disclosed