SCHEMBL6874286

SCHEMBL6874286

O=C(Nc1cccc(O)c1)c1ccc(C(=O)N[C@@H](Cc2ccc(NC(=O)c3c(Cl)cccc3Cl)cc2)C(=O)O)c(Cl)c1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.81
ITGA4 P13612 20/20 0.81
ITGA2 P17301 1/20 0.60
ITGB7 P26010 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6634573 0.90 ITGB1 (0.66) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6642500 0.90 ITGB1 (0.75) ITGB1ITGA4ITGA2ITGB7
SCHEMBL27682872 0.90 ITGB1 (0.75) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6642706 0.83 ITGB1 (0.80) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6637399 0.81 ITGB1 (0.72) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6641695 0.79 ITGB1 (0.80) ITGB1ITGA4ITGA2ITGB7
SCHEMBL18068435 0.79 ITGB1 (0.63) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15140174 0.78 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15145485 0.78 ITGB1 (0.60) ITGB1ITGA4ITGA2ITGB7
SCHEMBL15140177 0.78 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1403247-A1 N-Alkanoylphenylalanine derivatives F.HOFFMANN-LA ROCHE AG (CH) 2004-03-31 EP disclosed
US-6229011-B1 BINDING INHIBITORS BETWEEN VASCULAR ADHESION MOLECULE-1 AND ALPHA. BETA.INTEGRIN; USEFUL FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES SUCH AS MULTIPLE SCLEROSIS, ASTHMA, AND INFLAMMATORY BOWEL DISEASE HOFFMAN-LA ROCHE INC. 2001-05-08 US disclosed