SCHEMBL6635191

SCHEMBL6635191

CCOC(=O)Cn1c(COc2ccc(C(=N)N)cc2)nc2ccc(N(CCN(C)C)S(=O)(=O)c3ccccc3)cc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F2 P00734 8/20 0.44
F10 P00742 11/20 0.40
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
NPC1 O15118 1/20 0.37
NLRP3 Q96P20 1/20 0.37
PDE10A Q9Y233 1/20 0.37
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
NQO2 P16083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637038 0.94 F2 (0.49) F2F10MAPTNPSR1NPC1
SCHEMBL6640166 0.91 F2 (0.42) F2F10MAPTNPSR1NPC1
SCHEMBL6634421 0.89 HCRTR2 (0.39) MAPTNPSR1NPC1NLRP3
SCHEMBL6634703 0.86 F2 (0.53) F2F10
SCHEMBL6635194 0.85 F2 (0.39) F2F10NPSR1
SCHEMBL6636381 0.85 F2 (0.47) F2F10MAPTNPSR1NPC1
Hydrochloric Acid SCHEMBL8032330 0.84 F2 (0.57) F2F10
SCHEMBL6636049 0.83 F2 (0.57) F2F10PDE10AITGB3ITGA2B
SCHEMBL6642043 0.83 F2 (0.47) F2F10PDE10A
SCHEMBL6639197 0.83 MAPT (0.42) F2MAPTNPSR1NPC1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed