SCHEMBL6635205

SCHEMBL6635205

CC(=O)OCCOc1cccc(-c2c(NC(=O)Nc3c(C(C)C)cccc3C(C)C)c(=O)n(C)c3ncccc23)c1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACAT1 P24752 1/20 0.60
SOAT1 P35610 2/20 0.59
PDE4A P27815 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6634019 0.96 ACAT1 (0.61) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6635950 0.92 ACAT1 (0.68) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6634285 0.90 ACAT1 (0.72) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6634517 0.90 ACAT1 (0.76) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6634199 0.88 ACAT1 (0.61) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6635347 0.88 SOAT1 (0.66) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6633503 0.88 ACAT1 (0.57) ACAT1SOAT1
SCHEMBL6634432 0.88 ACAT1 (0.61) ACAT1SOAT1PDE4AKCNH2
SCHEMBL6636527 0.87 ACAT1 (0.58) ACAT1SOAT1
SCHEMBL6635775 0.86 ACAT1 (0.76) ACAT1SOAT1PDE4AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842933-B1 NOVEL NAPHTHYRIDINE DERIVATIVES SUMITOMO PHARMA (JP) 2004-08-04 EP disclosed
US-5843957-A Naphthyridine derivatives SUMITOMO PHARMACEUTICALS COMPANY, LTD. (JP) 1998-12-01 US disclosed
EP-0842933-A1 NOVEL NAPHTHYRIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-05-20 EP disclosed