SCHEMBL6636057

SCHEMBL6636057

CCOC(=O)CN(c1ccc2c(c1)nc(COc1ccc(C#N)cc1)n2CC)S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 5/20 0.57
MAPT P10636 6/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NPC1 O15118 3/20 0.44
NLRP3 Q96P20 1/20 0.44
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 3/20 0.38
TSHR P16473 1/20 0.38
ALOX5AP P20292 1/20 0.38
ATM Q13315 1/20 0.38
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
PGGT1B P53609 1/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6639246 0.93 F2 (0.67) F2MAPTNPSR1SMN1; SMN2GAA
SCHEMBL6639498 0.91 F2 (0.56) F2MAPTNPC1HTTHSD17B10
SCHEMBL6637177 0.90 F2 (0.72) F2MAPTNPSR1NPC1NLRP3
SCHEMBL6634298 0.86 F2 (0.61) F2MAPTNPSR1SMN1; SMN2GAA
SCHEMBL8138889 0.86 F2 (0.64) F2MAPTSMN1; SMN2GAATSHR
SCHEMBL8101459 0.86 F2 (0.68) F2MAPTSMN1; SMN2GAAFNTA
SCHEMBL6638786 0.85 F2 (0.65) F2MAPTSMN1; SMN2GAATSHR
SCHEMBL8109662 0.84 F2 (0.47) F2MAPTSMN1; SMN2GAATSHR
SCHEMBL6634546 0.84 F2 (0.47) F2MAPTNPC1HTTSMN1; SMN2
SCHEMBL6635659 0.84 F2 (0.54) F2HTTHSD17B10SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed