SCHEMBL663630

SCHEMBL663630

C=CCn1cc(C)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.51
MEN1 O00255 7/20 0.51
RAB9A P51151 2/20 0.50
NPC1 O15118 1/20 0.50
USP2 O75604 1/20 0.50
PDE4B Q07343 1/20 0.48
PDE4D Q08499 1/20 0.48
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
MAPT P10636 3/20 0.43
ALDH1A1 P00352 2/20 0.43
ALOX5 P09917 1/20 0.41
PRMT5 O14744 1/20 0.41
GSK3B P49841 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27418836 0.81 MEN1 (0.51) KMT2AMEN1RAB9ANPC1HDAC1
SCHEMBL8527697 0.81 MEN1 (0.55) KMT2AMEN1RAB9ANPC1HDAC1
SCHEMBL4520729 0.81 MEN1 (0.54) KMT2AMEN1RAB9ANPC1HDAC1
SCHEMBL8088590 0.79 MEN1 (0.51) KMT2AMEN1RAB9ANPC1USP2
SCHEMBL665932 0.79 MEN1 (0.56) KMT2AMEN1RAB9ANPC1USP2
SCHEMBL20054193 0.78 MEN1 (0.51) KMT2AMEN1RAB9ANPC1HDAC1
SCHEMBL4916450 0.78 MEN1 (0.48) KMT2AMEN1RAB9ANPC1USP2
SCHEMBL20931418 0.78 KMT2A (0.62) KMT2AMEN1RAB9ANPC1USP2
SCHEMBL15303762 0.78 MEN1 (0.48) KMT2AMEN1RAB9ANPC1USP2
SCHEMBL11130003 0.77 MEN1 (0.47) KMT2AMEN1RAB9ANPC1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116924964-A Preparation method of tetrahydrocarbazole ring compound 四川轻化工大学 2023-10-24 CN claimed
US-6391917-B1 ANALGESIC ZYMOGENETICS, INC. 2002-05-21 US claimed
US-6255351-B1 TREATMENT OF BONE DISORDERS ZYMOGENETICS, INC. 2001-07-03 US claimed
US-6221913-B1 Dialkyl ureas as calcitonin mimetics ZYMOGENETICS, INC. 2001-04-24 US claimed
US-6143932-A FOR EFFECTING ANALGESIA, A DECREASE IN THE POSTPRANDIAL RISE IN THE BLOOD GLUCOSE LEVELS OF A MAMMAL AFTER INGESTION OF A CARBOHYDRATE LOAD BY SAID MAMMAL, AND TREATING MICROBIAL INFECTIONS TREGA BIOSCIENCES, INC. (US) 2000-11-07 US claimed
EP-0975589-A2 DIALKYL UREAS AS CALCITONIN MIMETICS ZymoGenetics, Inc. (US) 2000-02-02 EP claimed
WO-1999037604-A2 DIALKYL UREAS AS CALCITONIN MIMETICS ZYMOGENETICS, INC. (US) 1999-07-29 WO claimed
US-5859190-A SOLID PHASE SYNTHESIS TO FORM A PROTECTED DIPEPTIDE FOLLOWED BY REACTING WITH 1,1'-THIOCARBONYLDIIMIDAZOLE TO EFFECT RING FORMATION; EFFICIENCY; ANTICONVULSANT,-ARRHYTHMIC AND DIABETIC AGENTS; HERBICIDES AND FUNGICIDES TREGA BIOSCIENCES, INC. (US) 1999-01-12 US claimed
WO-1998033776-A1 COMBINATORIAL LIBRARIES OF HYDANTOIN AND THIOHYDANTOIN DERIVATIVES, METHODS OF MAKING THE LIBRARIES AND COMPOUNDS THEREIN TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO claimed
CN-116924964-A Preparation method of tetrahydrocarbazole ring compound 四川轻化工大学 2023-10-24 CN disclosed
EP-3733428-B1 FUNCTIONALIZED ALUMINUM REAGENTS, METHOD OF MAKING A FUNCTIONALIZED ELASTOMER, ELASTOMER, RUBBER COMPOSITION AND TIRE GOODYEAR TIRE & RUBBER (US) 2022-03-16 EP disclosed
EP-3733428-A1 FUNCTIONALIZED ALUMINUM REAGENTS, METHOD OF MAKING A FUNCTIONALIZED ELASTOMER, ELASTOMER, RUBBER COMPOSITION AND TIRE The Goodyear Tire & Rubber Company (US) 2020-11-04 EP disclosed
US-10711016-B1 Functionalized aluminum reagents THE GOODYEAR TIRE & RUBBER COMPANY (US) 2020-07-14 US disclosed
CN-108101830-B A kind of 3- replaces the preparation method of Oxoindole and derivative 中国科学院成都生物研究所 2019-08-23 CN disclosed
US-6143932-A FOR EFFECTING ANALGESIA, A DECREASE IN THE POSTPRANDIAL RISE IN THE BLOOD GLUCOSE LEVELS OF A MAMMAL AFTER INGESTION OF A CARBOHYDRATE LOAD BY SAID MAMMAL, AND TREATING MICROBIAL INFECTIONS TREGA BIOSCIENCES, INC. (US) 2000-11-07 US disclosed
US-6121489-A Selectively N-alkylated peptidomimetic combinatorial libraries and compounds therein TREGA BIOSCIENCES, INC. (US) 2000-09-19 US disclosed
EP-0975589-A2 DIALKYL UREAS AS CALCITONIN MIMETICS ZymoGenetics, Inc. (US) 2000-02-02 EP disclosed
WO-1999037604-A2 DIALKYL UREAS AS CALCITONIN MIMETICS ZYMOGENETICS, INC. (US) 1999-07-29 WO disclosed
US-5859190-A SOLID PHASE SYNTHESIS TO FORM A PROTECTED DIPEPTIDE FOLLOWED BY REACTING WITH 1,1'-THIOCARBONYLDIIMIDAZOLE TO EFFECT RING FORMATION; EFFICIENCY; ANTICONVULSANT,-ARRHYTHMIC AND DIABETIC AGENTS; HERBICIDES AND FUNGICIDES TREGA BIOSCIENCES, INC. (US) 1999-01-12 US disclosed
WO-1998033776-A1 COMBINATORIAL LIBRARIES OF HYDANTOIN AND THIOHYDANTOIN DERIVATIVES, METHODS OF MAKING THE LIBRARIES AND COMPOUNDS THEREIN TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10711016-B1 Functionalized aluminum reagents C3AR1, FCGRT, ALK KMT2A 397/4885MEN1 318/4885RAB9A 1574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.