SCHEMBL6636734

SCHEMBL6636734

O=C(NNC(=O)c1cc2ccccc2cc1O)c1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 13/20 0.77
MEN1 O00255 10/20 0.77
POLB P06746 8/20 0.77
MAPT P10636 4/20 0.62
GAA P10253 3/20 0.62
TDP1 Q9NUW8 2/20 0.62
MITF O75030 1/20 0.62
NCOA1 Q15788 1/20 0.62
NCOA3 Q9Y6Q9 1/20 0.62
NPC1 O15118 2/20 0.61
RAB9A P51151 2/20 0.61
KDM4E B2RXH2 3/20 0.58
MAPK1 P28482 2/20 0.58
LMNA P02545 1/20 0.58
THRB P10828 1/20 0.58
MMP14 P50281 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
ALPL P05186 1/20 0.57
ALPI P09923 1/20 0.57
ALPG P10696 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13345885 0.91 KMT2A (0.73) KMT2AMEN1POLBMAPTGAA
SCHEMBL12857694 0.85 MEN1 (0.80) KMT2AMEN1POLBMAPTGAA
SCHEMBL13345883 0.84 KMT2A (0.65) KMT2AMEN1POLBMAPTGAA
SCHEMBL10597427 0.82 KMT2A (0.73) KMT2AMEN1POLBMAPTGAA
SCHEMBL4230145 0.80 KMT2A (0.63) KMT2AMEN1POLBMAPTGAA
SCHEMBL20536621 0.80 ALDH1A1 (0.58) KMT2AMEN1POLBMAPTGAA
SCHEMBL31354441 0.78 MEN1 (0.70) KMT2AMEN1POLBMAPTGAA
SCHEMBL5989960 0.78 KMT2A (0.61) KMT2AMEN1POLBMAPTGAA
SCHEMBL6638020 0.78 NPC1 (0.74) KMT2AMEN1GAANPC1RAB9A
SCHEMBL10724443 0.78 MEN1 (0.70) KMT2AMEN1POLBMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110034472-A1 Novel Compounds for Treatment of Cancer and Disorders Associated With Angiogenesis Function UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2011-02-10 US disclosed
US-20100120781-A1 Novel Compounds for Treatment of Cancer and Disorders Associated with Angiogenesis Function UNIVERSITY OF SOUTHERN CALIFORNIA 2010-05-13 US disclosed
US-20090093489-A1 NOVEL COMPOUNDS FOR TREATMENT OF CANCER AND DISORDERS ASSOCIATED WITH ANGIOGENESIS FUNCTION UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2009-04-09 US disclosed
EP-1420044-A2 Rubber composition and pneumatic tire Bridgestone Corporation (JP) 2004-05-19 EP disclosed
US-6380288-B1 LOW HEAT GENERATION PROPERTY, AGING REISTANCE, ALSO FOR PRODUCING VIBRATION ISOLATORS, BELTS AND HOSES AS WELL AS TIRE MATERIALS SUCH AS TIRE TREADS, UNDERTREADS, CARCASSES, SIDE WALLS AND BEADS BRIDGESTONE CORPORATION 2002-04-30 US disclosed
EP-0909788-A1 RUBBER COMPOSITION AND PNEUMATIC TIRES Bridgestone Corporation (JP) 1999-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034472-A1 Novel Compounds for Treatment of Cancer and Disorders Associated With Angiogenesis Function VEGFA, TEK, MCL1 KMT2A 3993/4885MEN1 2560/4885POLB 317/4885
US-20090093489-A1 NOVEL COMPOUNDS FOR TREATMENT OF CANCER AND DISORDERS ASSOCIATED WITH ANGIOGENESIS FUNCTION VEGFA, TEK, MCL1 KMT2A 3993/4885MEN1 2560/4885POLB 317/4885
US-20100120781-A1 Novel Compounds for Treatment of Cancer and Disorders Associated with Angiogenesis Function VEGFA, TEK, MCL1 KMT2A 3993/4885MEN1 2560/4885POLB 317/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.