SCHEMBL6637767

SCHEMBL6637767

Cn1c(CCc2ccc(C#N)cc2)nc2ncc(NS(=O)(=O)c3cccc4cccnc34)cc21

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.49
PKLR P30613 2/20 0.44
KMT2A Q03164 5/20 0.42
MEN1 O00255 4/20 0.42
GLO1 Q04760 1/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
BRD4 O60885 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633880 0.87 F2 (0.49) F2PKLRKMT2AMEN1GLO1
Hydrochloric Acid SCHEMBL6638514 0.85 F2 (0.67) F2PKLRKMT2AMEN1ALDH1A1
SCHEMBL6633872 0.82 F2 (0.50) F2PKLRKMT2AMEN1TP53
SCHEMBL8026354 0.80 F2 (0.74) F2PKLRKMT2AMEN1TP53
SCHEMBL8026334 0.77 F2 (0.55) F2PKLRKMT2AMEN1TP53
SCHEMBL6634709 0.76 F2 (0.57) F2PKLRKMT2AMEN1GLO1
SCHEMBL6636395 0.75 F2 (0.58) F2PKLRKMT2AMEN1GLO1
SCHEMBL6634125 0.75 F2 (0.58) F2PKLRKMT2AMEN1GLO1
SCHEMBL7985209 0.75 F2 (0.60) F2PKLRKMT2AMEN1TP53
SCHEMBL8029757 0.74 F2 (0.55) F2PKLRKMT2AMEN1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed