SCHEMBL6633880

SCHEMBL6633880

Cn1c(CCc2ccc(C#N)cc2)nc2cc(NS(=O)(=O)c3cccc4cccnc34)cnc21

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.49
PKLR P30613 2/20 0.44
GLO1 Q04760 2/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
SLC40A1 Q9NP59 2/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
POLB P06746 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
BRD4 O60885 1/20 0.41
ALPL P05186 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637767 0.87 F2 (0.49) F2PKLRGLO1KMT2AMEN1
Hydrochloric Acid SCHEMBL6637001 0.85 F2 (0.67) F2PKLRPKMKMT2AMEN1
SCHEMBL8026354 0.80 F2 (0.74) F2PKLRPKMKMT2AMEN1
SCHEMBL6633872 0.78 F2 (0.50) F2PKLRPKMKMT2AMEN1
SCHEMBL6634709 0.78 F2 (0.57) F2PKLRGLO1PKMKMT2A
SCHEMBL6638848 0.77 F2 (0.52) F2TP53ALDH1A1GAA
SCHEMBL6635303 0.76 PKM (0.51) F2PKLRGLO1PKMKMT2A
SCHEMBL7985209 0.75 F2 (0.60) F2PKLRPKMKMT2AMEN1
SCHEMBL6634125 0.75 F2 (0.58) F2PKLRGLO1PKMKMT2A
SCHEMBL6636395 0.75 F2 (0.58) F2PKLRGLO1PKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed