SCHEMBL6639262

SCHEMBL6639262

Cc1noc(NS(=O)(=O)c2ccccc2-c2ccc(-c3ccon3)cc2)c1C

nearest known ligand 0.75

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 10/20 0.75
EDNRB P24530 7/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777867 0.86 EDNRA (0.86) EDNRAEDNRB
SCHEMBL6151288 0.86 EDNRA (1.00) EDNRAEDNRB
SCHEMBL7948221 0.85 EDNRA (1.00) EDNRAEDNRB
SCHEMBL6767488 0.85 EDNRA (0.80) EDNRAEDNRB
SCHEMBL7956742 0.83 EDNRA (0.77) EDNRAEDNRB
SCHEMBL7947185 0.83 EDNRA (1.00) EDNRAEDNRB
SCHEMBL6640821 0.83 EDNRA (1.00) EDNRAEDNRB
SCHEMBL6641232 0.83 EDNRA (1.00) EDNRAEDNRB
SCHEMBL6772221 0.82 EDNRA (0.75) EDNRAEDNRB
SCHEMBL6772703 0.82 EDNRA (0.78) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702012-B1 Substituted isoxazole sulfonamides and their use as endothelin antagonists BRISTOL MYERS SQUIBB CO (US) 2003-10-15 EP claimed
US-5612359-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-18 US claimed
EP-0702012-A1 Substituted isoxazole sulfonamides and their use as endothelin antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-20 EP claimed
EP-0921800-B1 SUBSTITUTED BIPHENYL ISOXAZOLE SULFONAMIDES BRISTOL MYERS SQUIBB CO (US) 2004-04-14 EP disclosed
EP-0702012-B1 Substituted isoxazole sulfonamides and their use as endothelin antagonists BRISTOL MYERS SQUIBB CO (US) 2003-10-15 EP disclosed
US-5846990-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB CO. (US) 1998-12-08 US disclosed
US-5827869-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB COMPANY (US) 1998-10-27 US disclosed
US-5612359-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-18 US disclosed
EP-0702012-A1 Substituted isoxazole sulfonamides and their use as endothelin antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-20 EP disclosed