SCHEMBL6639670

SCHEMBL6639670

NC1=Nc2cc(C#Cc3ccccc3)ccc2C2CCCC12

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 20/20 0.60
NOS3 P29474 18/20 0.60
NOS2 P35228 18/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646269 0.82 NOS1 (0.79) NOS1NOS3NOS2
SCHEMBL6644831 0.76 NOS1 (1.00) NOS1NOS3NOS2
SCHEMBL6642386 0.76 NOS1 (0.60) NOS1NOS3NOS2
SCHEMBL6643582 0.76 NOS1 (0.69) NOS1NOS3NOS2
SCHEMBL6642383 0.76 NOS1 (0.60) NOS1NOS3NOS2
SCHEMBL6645211 0.74 NOS1 (1.00) NOS1NOS3NOS2
SCHEMBL6643807 0.74 NOS1 (1.00) NOS1NOS3NOS2
SCHEMBL6645947 0.74 NOS1 (0.68) NOS1NOS3NOS2
SCHEMBL6643315 0.73 NOS1 (1.00) NOS1NOS3NOS2
SCHEMBL6646529 0.70 NOS1 (0.67) NOS1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6391887-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE; CARDIOVASCULAR DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2002-05-21 US claimed
EP-1054869-B1 3,4-DIHYDROQUINOLINE DERIVATIVES AS NITROGEN MONOXIDE SYNTHASE (NOS) INHIBITORS SCHERING AG (DE) 2004-09-22 EP disclosed
US-6391887-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE; CARDIOVASCULAR DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2002-05-21 US disclosed